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Design, Synthesis and Antimicrobial Evaluation of New N-(1-Hydroxy-1,3-dihydrobenzo[c][1,2]oxaborol-6-yl)(hetero)aryl-2-carboxamides as Potential Inhibitors of Mycobacterial Leucyl-tRNA Synthetase |
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| Petr Šlechta, Adam Anthony Needle, Ondrej Jand’ourek, Pavla Paterová, Klára Konecná, Pavel Bárta, Jirí Kuneš, Vladimír Kubícek, Martin Doležal, Marta Kucerová-Chlupácová |
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In Vitro Antimycobacterial Activity of Human Lactoferrin-Derived Peptide, D-hLF 1-11, against Susceptible and Drug-Resistant Mycobacterium tuberculosis and Its Synergistic Effect with Rifampicin |
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| Sorasak Intorasoot, Amornrat Intorasoot, Arocha Tawteamwong, Bordin Butr-Indr, Ponrut Phunpae, Chayada Sitthidet Tharinjaroen, Usanee Wattananandkul, Sirikwan Sangboonruang, Jiaranai Khantipongse |
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Cyclic-di-AMP Phosphodiesterase Elicits Protective Immune Responses Against Mycobacterium tuberculosis H37Ra Infection in Mice |
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| Yanzhi Lu, Huanhuan Ning, Jian Kang, Guangchun Bai, Lei Zhou, Yali Kang, Zhengfeng Wu, Maolin Tian, Junhao Zhao, Yueyun Ma, Yinlan Bai |
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Hybridization Approach Toward Novel Antituberculars: Design, Synthesis, and Biological Evaluation of Compounds Combining Pyrazinamide and 4-Aminosalicylic Acid |
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A sensitive EZMTT method provides microscale, quantitative and high-throughput evaluation of drug efficacy in the treatment of Mycobacterium tuberculosis infectious diseases |
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| Li Xie,Zhao Chen,Wei Liu,Dongshi Gu,Yan Yu,Xinrou Chen,Yefei Wu,Ning Xu,Jie Xie,Gang Zhao,Benfang Helen Ruan |
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Improved solubility and stability of rifampicin as an inclusion complex of acyclic cucurbit[n]uril |
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Synthesis, Characterization and Biological Evaluation of New 3,5-Disubstituted-Pyrazoline Derivatives as Potential Anti-Mycobacterium tuberculosis H37Ra Compounds |
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Synthesis, Biological Evaluation, and In Silico Modeling of N-Substituted Quinoxaline-2-Carboxamides |
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Synthesis and Critical View on the Structure-Activity Relationships of N-(Substituted phenyl)-/N-Diphenylmethyl-piperazine-Based Conjugates as Antimycobacterial Agents |
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| Jana Curillová, Mária Pechácová, Tereza Padrtová, Daniel Pecher, Šárka Mascaretti, Josef Jampílek, Ludmila Pašková, František Bilka, Gustáv Kovác, Ivan Malík |
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| Martin Juhás,Lucie Kucerová,Ondrej Horácek,Ondrej Jandourek,Vladimír Kubícek,Klára Konecná,Radim Kucera,Pavel Bárta,Jirí Janoušek,Pavla Paterová,Jirí Kuneš,Martin Doležal,Jan Zitko |
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5-Alkylamino-N-phenylpyrazine-2-carboxamides: Design, Preparation, and Antimycobacterial Evaluation |
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| Weronika Ambrozkiewicz,Marta Kucerová-Chlupácová,Ondrej Jandourek,Klára Konecná,Pavla Paterová,Pavel Bárta,Jarmila Vinšová,Martin Doležal,Jan Zitko |
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| Qingwen Zhang,Jinxia Sun,Yan Fu,Weigang He,Yinhong Li,Hongsheng Tan,Hongxi Xu,Xin Jiang |
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